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BEAD BASED ASSAYS
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Aminodeoxychorismate Synthase Inhibitors from One-Bead One-Compound Combinatorial Libraries: “Staged” Inhibitor Design
Seth Dixon,† Kristin T. Ziebart,† Ze He,‡ Mellisa Jeddeloh,† Choong Leol Yoo,† Xiaobing Wang,§ Alan Lehman,§ Kit S. Lam, § Michael D. Toney,*,† and Mark J. Kurth*,†
†Department of Chemistry, University of California, One Shields Avenue, Davis, California 95616, ‡Department of Chemistry, Central Connecticut State University, 1615 Stanley Street, New Britain, Connecticut 06050, and §Department of Internal Medicine, Division of Hematology and Oncology, UC Davis Cancer Center, 4501 X Street, Sacramento, California 95817
J. Med. Chem., 49 (25), 7413 -7426, 2006. 10.1021/jm0609869 S0022-2623(06)00986-1
Web Release Date: November 10, 2006
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Biochemistry 45(1) pp 94 – 101 (2006) “SIRT1 Top 40 Hits: Use of One-Bead, One-Compound Acetyl-Peptide Libraries and Quantum Dots to Probe Deacetylase Specificity.”
Adam L. Garske and John M. Denu
Departments of Biomolecular Chemistry and Chemistry, University of Wisconsin, Madison, Wisconsin 53706
• DOI: 10.1021/bi052015l
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Organic Letters, Volume 6(21), Pages 3829-3832, “OBOC Small-Molecule Combinatorial Library Encoded by Halogenated Mass-Tags”
Sung Hee Hwang, Alan Lehman, Xin Cong, Marilyn M. Olmstead, Kit S. Lam, Carlito B. Lebrilla, and Mark J. Kurth
Department of Chemistry, University of California-Davis, One Shields Avenue, Davis, California 95616-5295, and Division of Hematology and Oncology, Department of Internal Medicine, University of California-Davis Cancer Center, 4501 X Street, Sacramento, California 95817
Web Release Date: September 17, 2004
• DOI: 10.1021/ol048408e
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QSAR & Combinatorial Science, Volume 22, Issue 7, Pages 754-766, "Solid Phase Combinatorial Library of 1,3-Azole Containing Peptides for the Discovery of Matrix Metallo Proteinase Inhibitors"
Caspar Christensen1, Christine Bruun Schiødt 2, Niels Tækker Foged2, Morten Meldal1 *,
1) Carlsberg Laboratory, Department of Chemistry, Gamle Carlsberg Vej 10, DK-2500 Valby, Denmark, 2) Nordic Bioscience A/S, Herlev Hovedgade 207, DK-2730 Herlev, Denmark.
Published Online 8 December 2003
• DOI: 10.1002/qsar.200320006
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J Comb Chem. 2004 May-Jun;6(3):312-24. "Combinatorial library of peptidotriazoles: identification of [1,2,3]-triazole inhibitors against a recombinant Leishmania mexicana cysteine protease."
Tornoe CW, Sanderson SJ, Mottram JC, Coombs GH, Meldal M. Center for Solid-Phase Organic Combinatorial Chemistry, Department of Chemistry, Carlsberg Laboratory, Gamle Carlsberg Vej 10, DK-2500 Valby, Denmark.
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18th American Peptide Symposium, July 19-23, 2003
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New Technology Automates Sorting of Large, Bead-based CombiChem Libraries, P127.
K. Ver Donck1, L. Bols1, R. Bongaarts1, P. Van Osta1, A. J. Brouwer2,
R. M. J. Liskamp2, D. Perrault3, K. Kalutkiewicz3, J. Geysen1, and R. Pulak3.
Union Biometrica-(Geel, BE1, Holliston, MA USA3), Utrecht University2 (Utrecht, NL).
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2nd European Symposium on Combinatorial Sciences (Eurocombi 2),
June 29-July 3
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From synthetic receptors towards synthetic antibodies using combinatorial chemistry, IN4.
Rob M.J. Liskamp, Arwin J. Brouwer, Christina Chamorro, Menno C.F. Monnee, Till Opatz, Roland J. Pieters, Dirk T.S. Rijkers, Kirk-Jan van Zoelen. Department of Medicinal Chemistry, Utrecht Institute for Pharmaceutical Sciences, Utrecht University, (Utrecht, The Netherlands).
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Protein affinity profiling using solid-phase combinatorial libraries, O19.
Anita J. Mathiesen, Sheryl Surve, Haifeng Yin, Phaedria M. St.Hilaire. Carlsberg Biosectro, Valby (Denmark).
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Bead-Based assays using COPAS™ Flow Sorting, P16.
K. Ver Donck1, L. Bols1, R. Bongaarts1, P. Van Osta1, A. J. Brouwer2,
R. M. J. Liskamp2, D. Perrault3, J. Geysen1, and R. Pulak3.
Union Biometrica-(Geel, BE1, Holliston, MA USA3), Utrecht University2 (Utrecht, NL).
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Innovative Combinatorial Approaches and Technologies, Practical Training Course (Florence, Italy) April 9-11, 2003
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Bead Based Assays Using COPAS Flow Sorting, Practical Session
R. Bongaarts and A. Comas. Union Biometrica, Geel, Belgium.
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Lab Automation 2003, February 1-5, 2003, Palm Springs, CA
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New technology automates sorting of large, bead--based combinatorial chemistry libraries, #87.
K. VerDonck1, L. Bols1, R. Bongaarts1, P. Van Osta1, J. Brouwer2, R. M. J. Liskamp2, J. Geysen1, D. Perrault3, K. Kalutkiewicz3, R. Pulak3 ~ Union Biometrica 1, 3, (Geel, BE 1; Holliston, MA 3), Utrecht University (Utrecht, NL 2)
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ISLAR 2002, October 20-23, 2002
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Assays for Bead-Based Technologies Using COPAS™ Flow Sorting, Session 3, Abstract 11.
K. Ver Donck1, L. Bols1, R. Bongaarts1, P. Van Osta1, A. J. Brouwer2, R. M. J. Liskamp2, J. Geysen1, D. Perrault3, K. Kalutkiewicz3, R. Pulak3, Union Biometrica-ESO 1, (Geel, BE), Union Biometrica 3, (Holliston, MA) Utrecht University 2 (Utrecht, NL)
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Biopolymers, 66(2) 93-100. "The one-bead two-compound assay for solid-phase screening of Combinatorial libraries."
Morton Meldal, Carlsberg Laboratory, Department of Chemistry, Gamle Carlsberg Vej 10,
DK-2500 Valby, Denmark.
SEPTEMBER, 2002
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MipTec-ICAR, May 27-30, 2002
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Optimizing the HTS Process: Assays beyond uHTS through COPAS™ Flow Sorting, #34.
K. Ver Donck, L. Bols, R. Bongaarts, P. Van Osta, A. J. Brouwer1, R. M. J. Liskamp1, J. Geysen,
Union Biometrica, 1) Utrecht University (Geel, BE; Utrecht, NL)
• View Abstract
• View updated Poster
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At the higher end of High Content Screening: The MIAS HTS imaging device, #82.
Kris Ver Donck, Luc Bols, Peter Van Osta, Johan Geysen, Union Biometrica, Cipalstraat 3, B-2440 Geel, Belgium
• View Abstract (PDF)
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Genetic Engineering News, Vol. 21, No. 20, November 15, 2001, "Firms Creating More Focused Compound Libraries, Saving Time and Money in Drug Discovery Research"
Author: Nina Flanagan.
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84th CSC Conference and Exhibition, May 2001
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Novel Methods for Analysis of Solid Phase Combinatorial Libraries on PEG-based Resins, #1134.
M. Meldal*, C. Gotfredsen, A. Papanikos, A. Meissner, M. Grotli, T. Groth, J. Beyer, J.
Duus, C. Tornoe, and P. St. Hilaire, SPOCC-center, Carlsberg Laboratory, Department of Chemistry,
Gamle Carlsberg Vej 10, DK-2500 Valby, Denmark.
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C = conference presentation
P = peer reviewed publication
A = printed periodical article
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